2015-2011

1.Straightforward Synthesis of Novel Enantiopure α-Trifluoromethylated Azetidine 2-Carboxylic Acid and Homoserines. Lensen, N.; Marais, J.; Brigaud, T. Org. Lett. 2015, 17, 342-345

2.Synthesis of Enantiopure trans-2,5-Disubstituted Trifluoromethylpyrrolidines and (2S,5R)‑5-Trifluoromethylproline. Lubin, H.; Pytkowicz, J.; Chaume, G.; Sizun-Thomé, G.; Brigaud, T. J. Org. Chem. 2015, 80, 2700-2708

3. Methionine sulfoxide- and sulfone-containing peptide synthesis: management of a relevant post-translational modification in proteins. Rentier, C.; Monasson, O.; Nuti, F.; Rovero, P.; Sabatino, G.; Papini, A-M. Chemistry Today 2015, 33, 32-36.

4. Synthesis of diastereomerically pure Lys(Nε-lipoyl) building blocks and their use in Fmoc/tBu solid phase synthesis of lipoyl-containing peptides for diagnosis of primary biliary cirrhosis. Rentier, C.; Pacini, G.; Nuti, F.; Peroni, E.; Rovero, P.; Papini, A-M. J. Pept. Sci. 2015, 21, 408-414.

5. Antibody Recognition in Multiple Sclerosis and Rett Syndrome Using a Collection of Linear and Cyclic N-glucosylated Antigenic Probes. Real Fernández, F.; Di Pisa, M.; Rossi, G.; Auberger, N.; Lequin, O.; Larregola, M.; Benchohra, A.; Mansuy, C.; Chassaing, G.; Lolli, F.; Hayek, J.; Lavielle, S.; Rovero, P.; Mallet, J-M.; Papini, A-M. Biopolymers 2015, 104, 560-576

6. Use of a (R)-α-Trifluoromethylalanine Containing Short Peptide in the Inhibition of Amyloid Peptide Fibrillation. Botz, A.; Gasparik, V.; Devillers, E.; Hoffmann, A. R. F.; Caillon, L.; Chelain, E.; Lequin, O.; Brigaud, T.; Khemtemourian, L. Biopolymers 2015, 104, 601-610

7. Role of lipoylation of the immunodominant epitope of pyruvate dehydrogenase complex: toward a peptide-based diagnostic immunoassay for primary biliary cirrhosis. Pacini, G.; Carotenuto, A.; Rentier, C.; Nuti, F.; Real-Fernandez, F.; Brancaccio, D.; Sabatino, G.; Larregola, M.; Peroni, E.; Migliorini, P.; Novellino, E.; Battezzati, P. M.; Selmi, C.; Papini, A. M.; Rovero, P. J. Med. Chem. 2015, 58, 6619-6629

8. Blanching of paint and varnish layers in easel paintings: contribution to the understanding of the alteration. Genty-Vincent, A.; Eveno, M.; Nowik, W.; Bastian, G.; Ravaud, E.; Cabillic, I.; Uziel, J.; Lubin-Germain, N.; Menu, M. Appl. Phys. A-Mater. 2015, 121, 779-788.

9. Interactions between Human Antibodies and Synthetic Conformational Peptide Epitopes: Innovative Approach for Electrochemical Detection of Biomarkers of Multiple Sclerosis at Platinum Electrodes. Bellagha-Chenchah, W.; Sella, C.; Real-Fernandez, F.; Peroni, E.; Lolli, F.; Amatore, C.; Thouin, L.; Papini, A. M. Electrochim. Acta 2015, 176, 1239-1247.

10. Synthesis of diastereomerically pure Lys(Nε-lipoyl) building blocks and their use in Fmoc/tBu solid phase synthesis of lipoyl-containing peptides for diagnosis of primary biliary cirrhosis. Rentier C., Pacini G., Nuti F., Peroni E., Rovero P., Papini A.M. J. Pept. Sci. 2015, 21, 408-414.

11. From the capillary condensation to the glass transition of a confined molecular liquid: Case of toluene. Audonnet, F.; Brodie-Linder, N.; Morineau, D.; Frick, B. J. Non-Cryst. Solids 2015, 407, 262-269.

12. Characterizing pigments with hyperspectral imaging variable false-color composites. Hayem-Ghez, A.; Ravaud, E.; Boust, C.; Bastian, G.; Menu, M.; Brodie-Linder, N. Appl. Phys. A 2015, 121, 939-947.

1. Copper(II) SBA-​15: A reusable catalyst for azide-​alkyne cycloaddition, Jlalia, I.; Gallier, F.; Brodie-Linder, N.; Uziel, J.; Auge, J.; Lubin-Germain, N. J. Mol. Catal. A: Chem. 2014, 393, 56-61.

2. Lubineau’s green synthons, Augé, J.; Lubin-Germain, N. Carbohydr. Chem. 2014, 40, 11-30.

3. Glaser oxidative coupling on peptides: Stabilization of β-turn structure via a 1,3-butadiyne constraint. Auberger, N.; Di Pisa, M.; Larregola, M.; Chassaing, G.; Peroni, E.; Lavielle, S.; Papini, A. -M.; Lequin, O.; Mallet, J. -M. Bioorg. Med. Chem. 2014, 22, 6924–6932.

4. 1,​4-​Disubstituted-​[1,​2,​3]​triazolyl-​Containing Analogues of MT-​II: Design, Synthesis, Conformational Analysis, and Biological Activity. Testa, C.; Scrima, M.; Grimaldi, M.; D'Ursi, A. M.; Dirain, M. L.; Lubin-Germain, N.; Singh, A.; Haskell-Luevano, C.; Chorev, M.; Rovero, P.; Papini, A. M. J. Med. Chem. 2014, 57, 9424-9434
.

5. New highlights on degradation process of verdigris from easel paintings. Santoro, C.; Zarkout, K.; Le Hô, A.S.; Mirambet, F.; Gourier, D.; Binet, L.; Pagès-Camagna, S.; Reguer, S.; Mirabaud, S.; Le Du, Y.; Griesmar, P.; Lubin-Germain, N.; Menu, M. Applied Physics A 2014. 114, 637-645.

1.Incorporation of CF₃−Pseudoprolines into Peptides: A Methodological Study. Chaume, G.; Simon, J.; Caupène, C.; Lensen, N.; Miclet, E.; Brigaud, T. J. Org. Chem. 2013, 78, 10144-10153.

2. Effects of enantiopure (S)-a-trifluoromethyl proline containing MIF-1’s analogue on stress-induced analgesia. Bocheva, A.; Nocheva, H.; Jlalia, I.; Lensen, N.; Chaume, G.; Brigaud, T. Med. Chem. 2013, 3, 206-209.

3.Synthesis of a MIF-1 analogue containing Enantiopure (S)-α-Trifluoromethyl Proline and Biological Evaluation on Nociception. Jlalia, I.; Lensen, N.; Chaume, G.; Dzhambazova, E.; Astasidi, L.; Hadjiolova, R.; Bocheva, A.; Brigaud, T. Eur. J. Med. Chem. 2013, 62, 122-129.

4. Conformational properties of peptides incorporating a fluorinated pseudoproline residue. Chaume, G.; Feytens, D.; Chassaing, G.; Lavielle, S.; Brigaud, T.; Miclet, E. New J. Chem. 2013, 37, 1336-1342.

5. Crystallization-Induced Dynamic Resolution of Fox Chiral Auxiliary and Application to the Diastereoselective Electrophilic Fluorination of Amide Enolates. Lubin, H.; Dupuis, C.; Pytkowicz, J.; Brigaud, T. J. Org. Chem. 2013, 78, 3487-3492.

6. Alpha actinin is specifically recognized by Multiple Sclerosis autoantibodies isolated using an N-glucosylated peptide epitope. Pandey, S.; Dioni, I.; Lambardi, D.; Real-Fernandez, F.; Peroni, E.; Pacini, G.; Lolli, F.; Seraglia, R.; Papini, A. M.; Rovero, P. Mol. Cell. Proteomics 2013, 12, 277–282.

7. Evaluation of new immunological targets in neuromyelitis optica. Chanson, J.-B.; Paolini, I.; Collongues, N.; Alcaro, M. C.; Blanc, F.; Barbetti, F.; Fleury, M.; Peroni, E.; Rovero, P.; Rudolf, G.; Lolli, F.; Trifilieff, É.; Papini, A.-M.; De Seze, J. J. Pept. Sci. 2013, 19, 25–32.

8. Method to create a hydrophilic environment within hydrophobic nanostructures, Brodie-Linder, N.; Deschamps, J.; Audonnet, F.; Alba-Simionesco, C. Micropor. Mesopor. Mat. 2013, 179, 17–21.

9. Total synthesis of high loading capacity PEG-based supports: evaluation and improvement of the process by use of ultrafiltration and PEG as a solvent, Turgis, R.; Billault, I.; Acherar, S.; Augé, J.; Scherrmann, M.-C. Green Chem. 2013, 15, 1016–1029.

1. Local control of the cis-trans isomerization and backbone dihedral angles in peptides using trifluoromethylated pseudoprolines, Feytens, D.; Chaume, G.; Chassaing, G.; Lavielle, S.; Brigaud, T.; Byun, B. J.; Kang, Y. K.; Miclet, E. J. Phys. Chem. B 2012, 116, 4069-4079.

2. Determination of the global material economy (GME) of synthesis sequences-a green chemistry metric to evaluate the greenness of products, Augé, J.; Scherrmann, M.-C. New J. Chem, 2012, 36, 1091-1098.

3. Straightforward glycosylation of alcohols and amino acids mediated by ionic liquid, Monasson, O.; Sizun-Thomé, G.; Lubin-Germain, N.; Uziel, J.; Augé, J. Carbohydr. Res. 2012, 352, 202-205

4. 2-Trifluoromethyl-2-methyl-4-phenyloxazolidine: A new chiral auxiliary for highly diastereoselective enolate alkylation, Tessier, A.; Pytkowicz, J.; Brigaud, T. J Fluorine Chem. 2012, 134, 122-127

5. Highly Diastereoselective Synthesis of Enantiopure β-Trifluoromethyl β-Amino Alcohols from Chiral Trifluoromethyl Oxazolidines (Fox), Simon, J.; Chelain, E.; Brigaud, T. Org. Lett., 2012, 14 (2), 604–607

6. Glycopeptide-Based Antibody Detection in Multiple Sclerosis by Surface Plasmon Resonance, Real-Fernandez, F.; Passalacqua, I.; Peroni, E.; Chelli, M.; Lolli, F.; Papini, A. M.; Rovero, P. Sensors 2012, 12, 5596-5607.

7. Designed glucopeptides mimetics of myelin protein epitopes as synthetic probes for the detection of autoantibodies, biomarkers of multiple sclerosis. Pandey, S.; Alcaro, M. C.; Scrima, M.; Peroni, E.; Paolini, I.; Di Marino, S.; Barbetti, F.; Carotenuto, A.; Novellino, E.; Papini, A. M.; D’Ursi, A. M.; Rovero, P. J. Med. Chem. 2012, 55, 10437–10447.

8. Alcohol to water catalyzed by Pt nanoparticles: an experimental and computational approach, Dehouche, F.; Archirel, P.; Remita, H.; Brodie-Linder, N.; Traverse, A.. RSC Advances 2012, 2, 6686.

9. Wall thickness determination of hydrophobically functionalized MCM-41 materials, Schoeffel, M.; Brodie-Linder, N.; Audonnet, F.; Alba-Simionesco, C. J. Mater. Chem. 2012, 22, 557–567.

1. Synthesis of trifluoromethyl cyclohexyl, cyclohexenyl and aryl compounds via stepwise Robinson annulation, Massicot, F.; Iriarte, A. M.; Brigaud, T.; Lebrun, A.; Portella, C. Org. Biomol. Chem. 2011, 2, 600-603.

2. Concise Synthesis of Enantiopure (S)- and (R)-alpha-Trifluoromethyl Aspartic Acid and alpha-Trifluoromethyl Serine from Chiral Trifluoromethyl Oxazolidines (Fox) via the Strecker-type Reaction, Simon, J.; Nguyen, T. T.; Chelain, E.; Lensen, N.; Pytkowicz, J.; Chaume, G.; Brigaud, T. Tetrahedron : Asymmetry 2011, 22, 309-314.

3. IgG and IgM antibodies to the refolded MOG(1-125) extracellular domain in humans, Gori, F.; Mulinacci, B.; Massai, L.; Avolio, C.; Caragnano, M.; Peroni, E.; Lori, S.; Chelli, M.; Papini, A-M.; Rovero, P. J. Neuroimmunol. 2011, 233, 216-220.

4. Titan Based Hybrid Organic-Inorganic Gels Comprising Carbohydrate Moiety, Danalev, D. L.; Lubin-Germain, N.; Serfaty, S.; Le Huerou, J-Y.; Auge, J.; Uziel, J.; Griesmar, P. Phosphorus Sulfur 2011, 186, 2216-2225.

5. La chimie verte pour un avenir plus rose, Augé, J.; Scherrmann, M.-C. Découverte 2011, 377, 28-37.